Pharmacokinetic parameters | Intravenous injection at a dose | Oral administration at doses | |
4.3 mg/kg | 4.3 mg/kg | 17.0 mg/kg | |
AUC (mg∙h/L) | 18.1 ± 1.5 | 14.2 ± 1.3 | 59.4 ± 6.1 |
fa (%) | 100.0 | 77.8 | 82.0 |