| Characteristics | Value |
| Gender ratio (male: female) | 1.06 (37:35) |
| Age (years)* | 38 ± 8.1 (21 - 57) |
| Body weight (kg)* | 49.7 ± 8.9 (30 - 68) |
| Baseline CD4 (cells/µL)¨ | 232 (6 - 716) |
| Baseline HIV-RNA (copies/mL)¨ | 91,318.5 (20 - 5,816,069) |
| Alanine transaminase (U/ml)¨ | 32.5 (5 - 126) |
| Aspartate transaminase (U/ml)¨ | 33 (11 - 248) |
| Total bilirubin (mg/dl)¨ | 0.3 (0.1 - 7.6) |
| CYP2B6 516G > T genotypes: |
|
| G/G carriers | 29 |
| G/T carriers | 29 |
| T/T carriers | 6 |