Entry | R1 | Oxaziridine Yield (%)a |
1 | Me (5) | 75 |
2 | n-Bu (6) | 68b |
3 | i-Bu (7) | 93 |
4 | tert-Bu (4) | 93 |
5 | Cy (8) | 69 |
6 | Ph (9) | 86 |
7 | 4-MeOC6H4 (10) | 79 |
8 | 4-NO2C6H4 (11) | 82 |