| α1 Subtype receptor selectivity | Drug name | Indication | |
| Hypertension | Benign prostatic hyperplasia | ||
| Non-selective |
|
|
|
|
| Prazosin | + | + |
|
| Bunazosin | + | ? |
|
| Terazosin | + | + |
|
| Urapidil | + | + |
|
| Doxazosin | + | ? |
| Selective |
|
|
|
|
| Naftopidil | ? | + |
|
| Silodosin | ? | + |
|
| Tamsulosin | ? | + |