Mechanisms | Drugs | References |
DNA Methyltransferase Inhibitors (DNMTi) | Azacytidine, Decitabine | [26] [100] |
Histone deacetylase inhibitors (HDACi) | Vorinostat, Belinostat Romidepsin, Panobinostat | [27] [103] [104] |
Histone methyltransferase inhibitors (HMTi) | 3-deazaneplanocin A (DZNep), Chaetocin | [28] [107] [108] |
Histone lysine methyltrasferase inhibitors (HLMi) | G9a, EZH2, GLP | [110] [111] |
Bromodomain and extra-terminal domain inhibitors (BETi) | JQ1, I-BET762 and OTX015 | [109] |
Epigenetic modulation of miRNA | Antisense Oligonucleotides (ASOs) | [29] |