Mechanisms

Drugs

References

DNA Methyltransferase Inhibitors (DNMTi)

Azacytidine, Decitabine

[26] [100]

Histone deacetylase inhibitors (HDACi)

Vorinostat, Belinostat Romidepsin, Panobinostat

[27] [103] [104]

Histone methyltransferase inhibitors (HMTi)

3-deazaneplanocin A (DZNep), Chaetocin

[28] [107] [108]

Histone lysine methyltrasferase inhibitors (HLMi)

G9a, EZH2, GLP

[110] [111]

Bromodomain and extra-terminal domain inhibitors (BETi)

JQ1, I-BET762 and OTX015

[109]

Epigenetic modulation of miRNA

Antisense Oligonucleotides (ASOs)

[29]