| Bioactivity | Active metabolite | Reference |
| Anti-tumor | Ganoderic acid S | Liu et al. (2009) |
| Ganoderic acid B | Hsu et al. (2008) | |
| Ganoderic acid F | Gao et al. (2006) | |
| Ganoderic acid Y | Jiang et al. (2011) | |
| Anti-HIV | Ganoderic acid B | Kang et al. (2015) |
| Ganoderic acid beta | Paydary et al. (2013) | |
| Anti-malaria | Ganoderic acid F | Lakornwong et al. (2014) |
| Schisanlactone B | Lakornwong et al. (2014) | |
| Ganoderiol F | Dondorp et al. (2009) | |
| Anti-hypertensive | Ganoderic acid K | Kabir et al. (1988) |
| Anti-hepatotoxic | Ganoderic acid R | Hirotani et al. (1986) |
| Hemostasis | Ganodermic acid S | Wang et al. (1989) |