| S. No. | Entry | R1 | R2 | R3 | 2 Yield (%) |
| 1 | a | H | HH | H | 80 |
| 2 | b | H | OH | H | 85 |
| 3 | c | OH | OH | H | 87 |
| 4 | d | H | OH | OH | 89 |