entry

catalyst

solvent

Temp/time

React medium/yielda

1

2

3

Bi(OTf)3, 10 mol%

Bi(OTf)3, 20 mol %

Bi(OTf)3, 30 mol %

EtOH

EtOH

EtOH

80˚C/6 h

80˚C/6 h

80˚C/6 h

One-pot, reflux/86%

One-pot, reflux/84%

One-pot, reflux/85%