|
| Pdb Code | Ligand | IC50 (nM) | Structure |
| 1 | 2A4L | R-roscovitine | 400 | Purine/Adenin Analogues Purine/Adenin Analogues Purine/Adenin Analogues |
| 2 | 1G5S | H717 | 48 | |
| 3 | 1W0X | OLOMOUCINE | 7 | |
| 4 | 1E1V | NU2058 | 17000 | O6-Substituted Guanines |
| 5 | 5D1J | BMs-387032/56H | 48 | Aminothiazole -based Inhibitors |
| 6 | 2BHE | 5-bromo Indirubin (BRY) | 80 | Oxindole-based Inhibitors |
| 7 | 1E1X | NU6027 (NW1) | 2200 | Aminopyrmidine Aminopyrmidine Aminopyrmidine |
| 8 | 1PXL | CK4 | 900 | |
| 9 | 3S2P | PMU | 68 | |
| 10 | 2R3Q | 5SC | 1 | Pyrazolopyrmidine Pyrazolopyrmidine |
| 11 | 3WBL | PDY | 23000 | |
| 12 | 2W05 | FRT | 1 | Imidazolopyrmidine |
| 13 | 1PXP | CK8 | 220 | Thiopyrmidine |
| 14 | 2VU3 | AT7519 | 47 | Pyrazolo based inhibitors Pyazolo based inhibitors |
| 15 | 2VTQ | LZA | 140 | |
| 16 | 2VV9 | IM9 | 17 | Triazole Based Inhibitors |