Patient

Targeted drugs (daily dose/duration)

PB

Pazopanib

Everolimus

Sirolimus

Dasatinib

Vorinostat

Erlotinib

Sorafenib

Lapatinib

Bevacizumab

Response

(date)

1

12 g/9 w

200 mg/1 w

400 mg/6 w

10 mg/ 3 w

200 mg/3 w

300 mg/ 8.5 w

150 mg/ 3 w

2.5 mg/kg × 1

5 mg/kg × 4

PR Nov 30, 2010

2

3 g/2 w

6 g/6 w

9 g/6 w

12 g/12 w

200 mg/9 w

1 mg/ 14 w

3 mg/ 2.5 w

50 mg/ 13 w

100 mg/ 12.5 w

SD May 17, 2012

4

12 g/ 7.3 w

200 mg/ 5.5 w

5 mg/ 6 w

50 mg/ 1 w

100 mg/ 5 w

10 mg/kg × 3

CR Apr 8, 2013

5

18 g/ 6 w

200 mg/1 w

400 mg/5 w

10 mg/ 6 w

750 mg/ 5.5 w

5 mg/kg × 1

10 mg/kg × 1

PR Jul 11, 2013

6

12 g/ 16 w

200 mg/ 15 w

10 mg/ 15.5 w

100 mg/6 w

150 mg/9.5 w

SD Feb 19, 2014

8

18 g/ 12 w

200 mg/ 6 w

5 mg/ 3 w

50 mg/ 7 w

10 mg/kg × 4

SD Sep 3, 2014

9

10 g/ 10 w

200 mg/ 3.5w

5 mg/ 9.5 w

50 mg/ 9.5 w

200 mg/ 5.5 w

8 mg/kg × 3

PR Aug 28, 2014

10

12 g/ 5.5 w

200 mg/ 5 w

5 mg/ 5.5 w

50 mg/ 4.5 w

10 mg/kg × 3

CR Sep 4, 2014

11

12 g/ 4 w

200 mg/ 4 w

5 mg/ 4 w

50 mg/ 3.5 w

10 mg/kg × 3

PR Sep 16, 2014