Compounds | CDK9 | CDK2 | |||
Ile25 | Phe30 | Val33 | Thr14 | Tyr15 | |
CAN508 | + | − | + | − | − |
NCI207113 | + | + | + | − | − |
TCM0004 | + | + | + | − | − |
TCM3282 | + | + | + | − | − |