Acetylcholine

Acetylthiocholine

Inhibitor (μmol/L)

kcat (s−1)

Km (μmol/L)

kcat/Km

(107 M−1 s −1)

Ki (μmol/L)

Inhibitor (μmol/L)

kcat (s−1)

Km (μmol/L)

kcat/Km

(107 M−1 s−1)

Ki (μmol/L)

0

11,315.2

138.3

8.18

9.72

0

9050.2

148.2

6.11

5.86

12.5

11,137.5

216.4

5.15

6.35

8661.1

205.9

4.21

25.0

11,101.5

663.8

1.67

10.0

8908.2

222.2

4.01

50.0

11,220.8

914.9

1.23

12.5

9024.0

475.1

1.90

75.0

11,180.1

1037.9

1.08

25.0

9088.3

916.5

0.99

--

--

--

--

50.0

9007.8

1087.0

0.83