| Drug class | Drug name |
| 4-aminoquinoline | Chloroquine (1) |
| Piperaquine (2) | |
| Amodiaquine (3) | |
| 8-aminoquinoline | Primaquine (4) |
| Quinine (5) | |
| Arylamino alcohol | Mefloquine (6) |
| Lumefantrine (9) | |
| Sesquiterpene lactone endoperoxides | Artemether (11) |
| Artesunate (12) | |
| Dihydroartemisinin (13) | |
| Mannich base | Pyronaridine(10) |
| Antifolate | Pyrimethamine (8) |
| Sulfadoxine (7) | |
| Proguanil (15) | |
| Naphthoquinone | Atovaquone (14) |