Structure/Name | Derivative | Target protein | ||
COX2 | NAT2 | TOP1 | ||
| D1 | −8.8 | −9.5 | −6.9 |
| D2 | −8.3 | −10.6 | −7.9 |
| D3 | −7.1 | −9.4 | −7.7 |
| D4 | −8.2 | −8.8 | −8 |
| D5 | −8.2 | −10.2 | −8.4 |
| D6 | −8.1 | −10.2 | −8.1 |