Drug

02

03

04

MW g/mol

360.36

486.56

500.58

TPSA (Å2)

110.62

116.69

116.69

(Consensus Log Po/w)

1.42

4.01

4.37

Lipinski rule

Yes

Yes

Yes

Bioactivity radar charts

Drug

05

06

07

MW g/mol

514.61

598.77

464.47

TPSA (Å2)

116.69

116.69

116.69

(Consensus Log Po/w)

4.78

6.93

3.10

Lipinski rule

Yes

No

Yes

Bioactivity radar charts