Drug | 02 | 03 | 04 |
MW g/mol | 360.36 | 486.56 | 500.58 |
TPSA (Å2) | 110.62 | 116.69 | 116.69 |
(Consensus Log Po/w) | 1.42 | 4.01 | 4.37 |
Lipinski rule | Yes | Yes | Yes |
Bioactivity radar charts |
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Drug | 05 | 06 | 07 |
MW g/mol | 514.61 | 598.77 | 464.47 |
TPSA (Å2) | 116.69 | 116.69 | 116.69 |
(Consensus Log Po/w) | 4.78 | 6.93 | 3.10 |
Lipinski rule | Yes | No | Yes |
Bioactivity radar charts |
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