No

LogP

MR

MV

IC₅₀ (AGS^*) (μM)

1

−0.35

65.36

177.7

75.2

2

0.11

70.19

193.9

82.1

3

0.75

94.59

240.6

2.5

4

0

96.47

239

15.5

5

0.7

101.26

264.6

2.8

6

1.19

94.58

244.8

3

7

0.64

101.26

264.6

4

8

0.71

94.58

244.8

5.2

9

0.95

107.94

288.6

9.1

10

0.88

99.29

259.1

2.1

11

1.42

103.92

275.6

3.9

12

0.99

87.57

242

2.5

13

0.33

87.02

237.9

4.6

14

1.46

94.77

256.2

NA**

15

2.28

109.17

284.8

2

16

1.21

99.41

256.9

1

17

0.46

101.29

255.3

3.3

18

1.16

106.09

280.9

5.5

19

1.65

99.4

261.1

1

20

1.66

105.96

268.7

1

21

1.1

106.09

280.9

>100

22

1.17

99.4

261.1

1.9

23

1.41

112.77

304.9

31.7

24

1.34

104.11

275.4

4.7

25

1.88

108.75

291.9

19.2

26

1.45

92.19

257.7

5.2

27

0.79

91.85

254.1

3.9

28

1.92

99.39

271.9

2.2

29

2.74

113.79

300.4

4.2