Reference

Temperature (˚C)

catalyst

solvent

Yield (%)

36

0

NaOH

H2O/Et2O

75

37

25

Lewis acid Y-Zr

MeCN

90

38

25

Zn

Benzene

97

40

25

Et3N

THF

43

41

10 - 15

NaOH

H2O

97

42

Reflux/IR

NaHCO3

Acetone

67.84