Parameters | Unit | Intravenous (10 mg/kg) | Oral (200 mg/kg) | ||
Mean | SD | Mean | SD | ||
AUC0−t | μg/mL*min | 1044.23 | 201.13 | 146 | 9.88 |
AUC0−∞ | μg/mL*min | 1131.45 | 159.52 | 325.33 | 69.73 |
MRT | h | 0.74 | 0.29 | 15.41 | 4.17 |
Tmax | min | 29.72 | 13.87 | / | / |
Cmax | ng/mL | 561.47 | 100.33 | / | / |
t1/2 | h | 0.85 | 0.19 | 10.47 | 3.25 |
AUMC0−∞ | H*h*ng/mL | 9589.94 | 1369.04 | 98857.22 | 43873.27 |
V | L/kg | 1.91 | 1.78 | 24.18 | 2.94 |
CL | L/h/kg | 0.92 | 0.3 | 1.68 | 0.41 |
Bioavailability, F | 0.69% |