Published IKr data only

Published & QPatch IKr data

QPatch IKr data only

Strong

Amiodarone

15a

99.99%

Pimozide

1a

99.0%

Astemizole

1a

1

97%

Azaperone

100

90%

Spiperone

47

90%

Bepridil

26b

99.8%

Risperidone

226a

90%

Clozapine

320h

670

95%

Loperamide

38

97%

Trifluperidol

20

90%

Clemastine

12c

96%

Tamoxifen

111xx

98%

Flunarizine

6i

120

99.97%

Methiothepin

140

99.2%

Triprolidine

340

90%

Dofetilide

5z

28%

Thioridazine

96a

99.0%

Fluspirilene

3a

1

99.87%

Naftopidil

190

99.1%

Domperidone

103a

92%

Trifluoperazine

234a

99.0%

Haloperidol

27h

25

92%

Naltriben

150

71%

Ifenprodil

88e

93%

Verapamil

136a

86%

Ketanserin

107a

120

95%

Naltrindole

220

76%

Lobeline

340f

76%

Vinpocetine

32a

66%

Mesoridazine

320h

490

95%

Nicergoline

56

95%

Pergolide

120a

98%

Terfenadine

11b

8

97%

Nifekalant

140

86%

Moderate

Amoxapine

1700j

90%

Metoclopramide

5400m

40%

Amlodipine

7800s

3100

99.5%

Alprenolol

6700

82%

Levallorphan

4900

35%

Chloroquine

2500a

57%

Mianserin

3200n

95%

Aripiprazole

1100j

470

99.0%

Benzamil

710

56%

Lofexidine

8500

85%

Chlorpromazine

370yy

94%

Miconazole

2100o

99.0%

Carvedilol

510d

540

98%

Benzydamine

1500

81%

Lomerizine

600

99.65%

Citalopram

950k

80%

Olanzapine

6000g

93%

Dextromethorphan

5100u

5700

55%

Bopindolol

1600

65%

Manidipine

940

99.0%

Desloratadine

6300l

85%

Prazosin

1600a

94%

Diltiazem

9100a

1100

82%

Butaclamol

490

98%

Naloxone

1800

46%

Diphenhydramine

2600a

81%

Promethazine

1500p

91%

Dolasetron

6000v

4100

72%

Cilnidipine

3100

99.88%

Naltrexone

6700

21%

Fluoxetine

460a

94%

Quetiapine

5800g

83%

Doxazosin

600a

390

98%

Cirazoline

6000

24%

Nicardipine

670

99.0%

Fluphenazine

997 j

90%

Raloxifene

1100q

99.4%

Escitalopram

2600oo

1100

46%

Cyclosporine

6700

93%

Niguldipine

710

99.6%

Imipramine

1900a

93%

Ranolazine

14,600a

0%

Flecainide

3900w

1600

48%

Cyproheptadine

1500

96%

Nimodipine

2100

98%

Ketoconazole

1900a

99.0%

Remoxipride

2300 j

84%

Granisetron

3700v

6700

65%

Dilazep

600

10%

Nisoxetine

850

97%

Loratadine

7900l

97%

Sibutramine

2500r

97%

Maprotiline

3100a

1500

89%

Disulfiram

2800

96%

Phenamil

1200

67%

Mepyramine

6000x

910

70%

Dorzolamide

7500

33%

Phentolamine

850

58%

Ondansetron

810v

850

73%

Felodipine

1800

99.6%

Quinacrine

1200

87%

Primaquine

2000y

6000

65%

Gestrinone

6000

97%

Strychnine

1200

60%

Propafenone

440w

370

96%

Harmine

1500

89%

Tacrine

910

75%

Propranolol

3900d

7500

87%

Hydroxytacrine

5700

53%

Telmisartan

2100

99.6%

Imiquimod

850

72%

Tropisetron

1800

71%

Lacidipine

1700

93%

Vinorelbine

6000

13%

Weak

Bupivacaine

20,000aa

94%

Propofol

36,000gg

98%

Capsaicin

17,450ee

41,000

97%

Betaxolol

15,000

60%

Zonisamide

18,000

Chlorpheniramine

13,000x

30%

Roxithromycin

37,000bb

15%

Nelfinavir

11,000ii

7500

98%

Denbufylline

13,000

52%

Clarithromycin

33,000bb

77%

Sildenafil

33,000hh

96%

Nifedipine

135,000s

4700

96%

Diazoxide

14,000

94%

Fluconazole

48,000cc

11%

Sparfloxacin

30,000a

45%

Nitrendipine

18,100s

1600

98%

Nalbuphine

16,000

50%

Glimepiride

74,000dd

99.5%

Spironolactone

23,000a

98%

Physostigmine

15,000

46%

Imatinib

20,000z

95%

Terazosin

17,000a

92%

Estradiol

>100,000kk

8000

98%

Pronethalol

13,000

73%

Lovastatin

12,500a

95%

Vardenafil

13,000hh

95%

Quinpirole

15,000

Nisoldipine

23,000ff

99.7%

Venlafaxine

28,000k

27%

Tramadol

16,000

20%