| Published IKr data only | Published & QPatch IKr data | QPatch IKr data only | |||||||||||||
Strong | Amiodarone | 15a | 99.99% | Pimozide | 1a | 99.0% | Astemizole | 1a | 1 | 97% | Azaperone | 100 | 90% | Spiperone | 47 | 90% |
Bepridil | 26b | 99.8% | Risperidone | 226a | 90% | Clozapine | 320h | 670 | 95% | Loperamide | 38 | 97% | Trifluperidol | 20 | 90% | |
Clemastine | 12c | 96% | Tamoxifen | 111xx | 98% | Flunarizine | 6i | 120 | 99.97% | Methiothepin | 140 | 99.2% | Triprolidine | 340 | 90% | |
Dofetilide | 5z | 28% | Thioridazine | 96a | 99.0% | Fluspirilene | 3a | 1 | 99.87% | Naftopidil | 190 | 99.1% |
|
|
| |
Domperidone | 103a | 92% | Trifluoperazine | 234a | 99.0% | Haloperidol | 27h | 25 | 92% | Naltriben | 150 | 71% |
|
|
| |
Ifenprodil | 88e | 93% | Verapamil | 136a | 86% | Ketanserin | 107a | 120 | 95% | Naltrindole | 220 | 76% |
|
|
| |
Lobeline | 340f | 76% | Vinpocetine | 32a | 66% | Mesoridazine | 320h | 490 | 95% | Nicergoline | 56 | 95% |
|
|
| |
Pergolide | 120a | 98% |
|
|
| Terfenadine | 11b | 8 | 97% | Nifekalant | 140 | 86% |
|
|
| |
Moderate | Amoxapine | 1700j | 90% | Metoclopramide | 5400m | 40% | Amlodipine | 7800s | 3100 | 99.5% | Alprenolol | 6700 | 82% | Levallorphan | 4900 | 35% |
Chloroquine | 2500a | 57% | Mianserin | 3200n | 95% | Aripiprazole | 1100j | 470 | 99.0% | Benzamil | 710 | 56% | Lofexidine | 8500 | 85% | |
Chlorpromazine | 370yy | 94% | Miconazole | 2100o | 99.0% | Carvedilol | 510d | 540 | 98% | Benzydamine | 1500 | 81% | Lomerizine | 600 | 99.65% | |
Citalopram | 950k | 80% | Olanzapine | 6000g | 93% | Dextromethorphan | 5100u | 5700 | 55% | Bopindolol | 1600 | 65% | Manidipine | 940 | 99.0% | |
Desloratadine | 6300l | 85% | Prazosin | 1600a | 94% | Diltiazem | 9100a | 1100 | 82% | Butaclamol | 490 | 98% | Naloxone | 1800 | 46% | |
Diphenhydramine | 2600a | 81% | Promethazine | 1500p | 91% | Dolasetron | 6000v | 4100 | 72% | Cilnidipine | 3100 | 99.88% | Naltrexone | 6700 | 21% | |
Fluoxetine | 460a | 94% | Quetiapine | 5800g | 83% | Doxazosin | 600a | 390 | 98% | Cirazoline | 6000 | 24% | Nicardipine | 670 | 99.0% | |
Fluphenazine | 997 j | 90% | Raloxifene | 1100q | 99.4% | Escitalopram | 2600oo | 1100 | 46% | Cyclosporine | 6700 | 93% | Niguldipine | 710 | 99.6% | |
Imipramine | 1900a | 93% | Ranolazine | 14,600a | 0% | Flecainide | 3900w | 1600 | 48% | Cyproheptadine | 1500 | 96% | Nimodipine | 2100 | 98% | |
Ketoconazole | 1900a | 99.0% | Remoxipride | 2300 j | 84% | Granisetron | 3700v | 6700 | 65% | Dilazep | 600 | 10% | Nisoxetine | 850 | 97% | |
Loratadine | 7900l | 97% | Sibutramine | 2500r | 97% | Maprotiline | 3100a | 1500 | 89% | Disulfiram | 2800 | 96% | Phenamil | 1200 | 67% | |
|
|
|
|
|
| Mepyramine | 6000x | 910 | 70% | Dorzolamide | 7500 | 33% | Phentolamine | 850 | 58% | |
|
|
|
|
|
| Ondansetron | 810v | 850 | 73% | Felodipine | 1800 | 99.6% | Quinacrine | 1200 | 87% | |
|
|
|
|
|
| Primaquine | 2000y | 6000 | 65% | Gestrinone | 6000 | 97% | Strychnine | 1200 | 60% | |
|
|
|
|
|
| Propafenone | 440w | 370 | 96% | Harmine | 1500 | 89% | Tacrine | 910 | 75% | |
|
|
|
|
|
| Propranolol | 3900d | 7500 | 87% | Hydroxytacrine | 5700 | 53% | Telmisartan | 2100 | 99.6% | |
|
|
|
|
|
|
|
|
|
| Imiquimod | 850 | 72% | Tropisetron | 1800 | 71% | |
|
|
|
|
|
|
|
|
|
| Lacidipine | 1700 | 93% | Vinorelbine | 6000 | 13% | |
Weak | Bupivacaine | 20,000aa | 94% | Propofol | 36,000gg | 98% | Capsaicin | 17,450ee | 41,000 | 97% | Betaxolol | 15,000 | 60% | Zonisamide | 18,000 |
|
Chlorpheniramine | 13,000x | 30% | Roxithromycin | 37,000bb | 15% | Nelfinavir | 11,000ii | 7500 | 98% | Denbufylline | 13,000 | 52% |
|
|
| |
Clarithromycin | 33,000bb | 77% | Sildenafil | 33,000hh | 96% | Nifedipine | 135,000s | 4700 | 96% | Diazoxide | 14,000 | 94% |
|
|
| |
Fluconazole | 48,000cc | 11% | Sparfloxacin | 30,000a | 45% | Nitrendipine | 18,100s | 1600 | 98% | Nalbuphine | 16,000 | 50% |
|
|
| |
Glimepiride | 74,000dd | 99.5% | Spironolactone | 23,000a | 98% |
|
|
|
| Physostigmine | 15,000 | 46% |
|
|
| |
Imatinib | 20,000z | 95% | Terazosin | 17,000a | 92% | Estradiol | >100,000kk | 8000 | 98% | Pronethalol | 13,000 | 73% |
|
|
| |
Lovastatin | 12,500a | 95% | Vardenafil | 13,000hh | 95% |
|
|
|
| Quinpirole | 15,000 |
|
|
|
| |
Nisoldipine | 23,000ff | 99.7% | Venlafaxine | 28,000k | 27% |
|
|
|
| Tramadol | 16,000 | 20% |
|
|
|