Biochemical profilinga | IC50 (nmol/l)b | Ki [ATP] (nmol/l)b |
CDK4/cyclin D1 | 2.0 ± 0.4 (n = 5) | 0.6 ± 0.3 (n = 2) |
CDK6/cyclin D1 | 9.9 (n = 1) | 2.4 ± 1.2 (n = 2) |
CDK1/cyclin B1 | 1627 ± 666 (n = 5) | - |
CDK2/cyclin E | 504 ± 298 (n = 3) | - |
CDK9/cyclin T1 | 57 ± 42 (n = 4) | - |
CDK7/Mat1/cyclin H1 | 3910 ± 2410 (n = 4) | - |
PIM1 | 50 (n = 1) | - |
PIM2 | 3400 (n = 1) | - |
ERK1 | >20,000 (n = 1) | - |