Compound

Cancer cell line

IC50 (μM)

Compound

Cancer cell line

IC50 (μM)

179a

T47D

13.2 ± 1.4

180a

Colo-829

1.13 ± 0.03

179a

A549

8.58 ± 1.70

180a

A549

1.62 ± 0.91

179b

A549

14.3 ± 0.3

180b

C-32

1.33 ± 0.12

181a

T47D

1.47 ± 0.32

180b

MDA-MB-231

5.88 ± 0.88

181b

SNB-19

3.38 ± 0.15

182a

A549

13.5 ± 1.5

181b

Colo-829

1.08 ± 0.06

182b

Colo-829

6.67 ± 1.30

181b

A549

1.15 ± 0.10

182b

C-32

1.27 ± 0.06

183a

Colo-829

4.68 ± 0.33

182b

MDA-MB-231

2.43 ± 0.68

183a

MCF-7

1.58 ± 0.17

182b

A549

0.45 ± 0.20

183a

MDA-MB-231

0.90 ± 0.01

183b

SNB-19

10.8 ± 0.5

183a

A549

0.59 ± 0.13

184a

SNB-19

7.54 ± 0.38

184a

Colo-829

0.13 ± 0.03

184b

C-32

1.04 ± 0.10

184a

C-32

1.72 ± 0.22

184b

MDA-MB-23

6.77 ± 0.85

184a

MCF-7

8.72 ± 0.47

184b

A549

1.28 ± 0.06

184a

T47D

12.31 ± 0.77

185a

Colo-829

0.13 ± 0.01

184a

A549

0.77 ± 0.12

185a

A549

3.30 ± 0.48

185b

Colo-829

0.12 ± 0.03

185b

MCF-7

0.94 ± 0.03

185b

C-32

1.14 ± 0.12

185b

MDA-MB-231

0.11 ± 0.01

185b

A549

0.84 ± 0.01