Inhibitors | 1'-hydroxymidazolam | 4-hydroxymidazolam | ||||
Vmax (nmol/min/kg) | Km (mM) | Ki (mM) | Vmax (nmol/min/kg) | Km (mM) | Ki (mM) | |
CPFX | 0.15 ± 0.06 | 14.62 ± 13.24 | 5.81 ± 5.48 | 0.15 ± 0.07 | 32.36 ± 16.86 | 9.13 ± 2.23 |
OBFX | 0.14 ± 0.08 | 15.76 ± 19.4 | 11.68 ± 3.45 | 0.11 ± 0.05 | 29.29 ±10.45 | 21.11 ± 11.92 |
NFX | 0.12 ± 0.07 | 5.07± 3.90 | 25.60 ± 12.94 | 0.13 ± 0.06 | 29.11 ± 14.01 | 24.11 ± 13.95 |
OFX | 0.17 ± 0.06 | 43.78 ± 50.76 | 32.98 ± 20.40 | 0.15 ± 0.08 | 39.43 ±17.22 | 23.05 ± 7.24 |
EFX | 0.14 ± 0.08 | 6.04 ± 6.27 | 34.68 ± 31.49 | 0.14 ± 0.09 | 29.88 ± 4.26 | 28.76 ± 14.67 |