48
R = 3-F, 5-F
O
47
+++
49
R = 3-F, 4-F, 5-F
O
91
+
50
R = 3-Me, 4-NO2
O
180
N/A
51
R = 3-Me, 4-NH2
O
600
N/A
52
R2 = 4-Et
O
190
N/A
53
R = 4-Prop
O
110
+
55
R = 4-OEt
O
56
+
61
R = 4-I
O
210
N/A
62
R = 4-NO2
O
>1000
N/A
64
R1 = 
-
330
N/A
65
R1 = 
-
100
+++
66
R1 = 
-
770
N/A
67
R1 = 
-
>1000
N/A
A8
R = H
NH
470
N/A
A10
R = 2-Et
NH
350
N/A
A12
R = 2-Me, 3-Me
NH
230
N/A
A17
R = 3-OMe
NH
120
+++
A21
R = 3-Me, 4-Me
NH
230
N/A
A23
R = 3-tBut, 5-tBut
NH
>1000
N/A
A25
R = 3-OMe, 4-OMe
NH
610
N/A
A26
R = 3-OMe, 5-OMe
NH
170
+++
A28
R = 4-Me
NH
610
N/A
A30
R = 4-But
NH
770
N/A
A31
R = 4-secBut
NH
>1000
N/A
A32
R = 4-tBut
NH
>1000
N/A
A35
R = 4-Hept
NH
>1000
N/A
A36
R = 4-OMe
NH
>1000
N/A
A39
R = 4-Br
NH
240
N/A
A40
R = 4-Cl
NH
170
N/A
A41
R = 4-F
NH
690
N/A
A42
R = 4-I
NH
600
N/A
A45
R1 = 
NH
460
N/A
A46
R1 = 
NH
480
N/A
A47
R1 = 
NH
240
N/A
A48
R1 = 
NH
170
++