Compound

R

Cell line

HT-29

HELA

A-549

FA1

H

20 ± 2

35 ± 2

18 ± 1

FA2

Methyl

55 ± 2

45 ± 1

40 ± 1

FA3

Ethyl

50 ± 1

NA

70 ± 2

FA4

Benzyl

38 ± 1

65 ± 2

50 ± 2

FA5

Aniline

90 ± 1

120 ± 2

NA

FA6

4-amino benztrifluoride

19 ± 2

38 ± 2

66 ± 1

FA7

Amino benz nitrile

NA

80 ± 2

72 ± 1

FA8

p-hydroxy aniline

50 ± 2

90 ± 1

40 ± 2

FA9

p-fluoro benzyl

30 ± 1

25 ± 2

55 ± 2

FA10

Morpholine

18 ± 2

23 ± 1

30 ± 1

Methotrexate

12 ± 1

9 ± 1

5 ± 1