Drug name | Antipsychotic class | CYPa isoform |
Known to prolong the QTc interval |
|
|
Bromperidol [51] | Typical | 3A4 [47] |
Chlorpromazine [26] [52] | Typical | 2D6 [38] |
Fluphenazine decanoate [53] [54] | Typical | 2D6 [50] |
Haloperidol [55] [56] | Typical | 2D6 [50] |
Haloperidol decanoate [52] [57] | Typical | 2D6 [34] [48] |
Levomepromazine [52] [58] | Typical | 2D6 [49] |
Nemonapride [59] | Typical | 2D6 [30] |
Olanzapine [60] [61] | Atypical | 1A2, 2D6 [45] |
Perphenazine [8] [40] | Typical | 2D6 [45] |
Pimozide [41] [62] | Typical | 1A2, 2D6, 3A4 [33] |
Quetiapine [42] [60] | Atypical | 3A4 [4] [35] |
Risperidone [60] [63] | Atypical | 2D6 [32] |
Trifluoperazine [64] | Typical | 1A2 [44] |
No available information on QTc interval |
|
|
Perospirone | Atypical | 1A2, 2C8, 2D6, 3A4 [5] |
Zotepine | Atypical | 1A2, 2B6, 2C9, 2C19, 2D6, 3A4, 3A5 [5] |