L882I

enzalutamide

LBD

[2]

unknown

S889G

bicalutamide,

enzalutamide

LBD

[48]

antagonist-to-agonist

switch

D891H

bicalutamide

LBD

[48]

antagonist-to-agonist

switch

E894K

enzalutamide

LBD

[2]

unknown

M896T/V

bicalutamide,

S-1

LBD

[1] [40] [48]

antagonist-to-agonist

switch