L882I | enzalutamide | LBD | [2] | unknown |
S889G | bicalutamide, enzalutamide | LBD | [48] | antagonist-to-agonist switch |
D891H | bicalutamide | LBD | [48] | antagonist-to-agonist switch |
E894K | enzalutamide | LBD | [2] | unknown |
M896T/V | bicalutamide, S-1 | LBD | [1] [40] [48] | antagonist-to-agonist switch |