| Acarbose | Neosalacinol | ||
Human | rat | Human | rat | |
NtMGAM | −1.5 | −15.4 | −20.6 | −20.6 |
NtSI | −4.3 | −2.0 | −12.5 | −27.6 |
CtMGAM | −8.3 | −13.3 | −23.6 | −7.0 |
CtSI | −12.5 | −12.4 | −14.1 | −13.9 |
Average of four domains | −6.7 | −10.9 | −17.7 | −17.3 |
IC50 (μM)a | 15.2 | 1.7 | 9.0 | 22.2 |